Peptide and Clinical Reference Library

What is Tirzepatide

Tirzepatide is a novel investigational dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist being developed for the treatment of type 2 diabetes. GIP and GLP-1 are hormones that play crucial roles in regulating blood sugar levels, insulin secretion, and appetite. Tirzepatide works by activating both GIP and GLP-1 receptors,leading to improved glycemic control, weight loss, and potentially cardiovascular benefits.

Clinical trials have shown promising results, with tirzepatide demonstrating superior efficacy compared to traditional GLP-1 receptor agonists in reducing HbA1c levels and body weight. If approved by regulatory authorities, tirzepatide has the potential to become a valuable addition to the armamentarium of diabetes treatments available to healthcare professionals for managing this chronic condition effectively.